Fig. 1 · Structure
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Apstatin
APP Inhibitor
Apstatin is a potent inhibitor of aminopeptidase P (APP), exhibiting Ki values of 2.6 µM for rat APP and 0.64 µM for human APP. This compound has demonstrated cardioprotective effects, making it a valuable tool for research into cardiovascular diseases and related pathologies. Its ability to modulate APP activity positions it as a significant reagent for studies focused on peptide metabolism and cardiac health.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 160470-73-5 |
| Applications | APP Inhibitor |
| Formula | C23H33N5O5 |
| Molecular Weight | 459.54 |
| SMILES | C[C@@H](C(N)=O)NC([C@H]1N(C([C@H]2N(C([C@@H](O)[C@H](N)CC3=CC=CC=C3)=O)CCC2)=O)CCC1)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.