ASTX-660

Catalog No.: A16996

XIAP inhibitor

ASTX-660

ASTX-660 Chemical Structure

CAS NO. 1799328-86-1

ASTX660 is an orally bioavailable, non-peptidomimetic antagonist of both X chromosome-linked inhibitor of apoptosis protein (XIAP) and cellular IAP 1 (cIAP1), with potential antineoplastic and pro-apoptoticctivities. 1799328-86-1 (free base) 1799328-50-9 (HCl) 1799328-90-7 (mesylate) 1799328-88-3 (sulfate)

Availability: In stock

Package Price Qty
1 mg
$380.00
2 mg
$600.00
5 mg
$1,200.00
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Biological Activity

ASTX660 is an orally bioavailable, non-peptidomimetic antagonist of both X chromosome-linked inhibitor of apoptosis protein (XIAP) and cellular IAP 1 (cIAP1), with potential antineoplastic and pro-apoptoticctivities. 1799328-86-1 (free base) 1799328-50-9 (HCl) 1799328-90-7 (mesylate) 1799328-88-3 (sulfate)
In vitro DMSO 93 mg/mL (172.32 mM)
Water 93 mg/mL (172.32 mM)
Ethanol Insoluble
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 18.53 mL 92.65 mL 185.29 mL
0.5 mM 3.71 mL 18.53 mL 37.06 mL
1 mM 1.85 mL 9.26 mL 18.53 mL
5 mM 0.37 mL 1.85 mL 3.71 mL

*The above data is based on the productmolecular weight 539.69. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A16996
Actions Inhibitor
CAS No. 1799328-86-1
Formula C30H42FN5O3
M. Wt 539.69
Solubility DMSO
Purity >98%
Synonyms ASTX660, ASTX 660
SMILES OCC1=NC2=C(N(CC2(C)C)C(CN3[[email protected]@H](CN4[[email protected]](C)COCC4)CN[[email protected]](C)C3)=O)C=C1CC5=CC=C(F)C=C5
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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