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AT1R antagonist 4

AT1R Antagonist

AT1R antagonist 4 is a selective antagonist of the angiotensin II type 1 receptor (AT1R). It demonstrates significant inhibitory activity on calcium influx in cells that stably express both AT1 and ETA receptors. This compound is particularly useful in kidney disease research, enabling investigations into the role of angiotensin signaling in renal pathophysiology.

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Specifications

Manufacturer	Adooq Bioscience
Actions	Antagonist
CAS Number	2982582-16-9
Applications	AT1R Antagonist
Formula	C₂₁H₁₆BrN₃O₅S
Molecular Weight	502.34
SMILES	O=C1NC(C2=C1C(Br)=CC=C2NS(=O)(C3=CC(C#CC4=NOC(C)=C4C)=CC=C3)=O)O

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.