Fig. 1 · Structure
Documents & Downloads
Axelopran sulfate
Opioid Receptor Antagonist
Axelopran sulfate is a potent opioid receptor antagonist, exhibiting pKi values of 9.8, 8.8, and 9.9 for human recombinant μ and δ opioid receptors, as well as the guinea pig κ receptor. This compound is valuable for research focused on opioid signaling mechanisms and may aid in the investigation of pain management and addiction pathways. Its activity makes it a useful tool for elucidating the role of opioid receptors in various biological processes.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 949904-50-1 |
| Applications | Opioid Receptor Antagonist |
| Formula | C26H41N3O8S |
| Molecular Weight | 555.68 |
| Synonyms | TD-1211 sulfate |
| SMILES | O=C([C@@H](O)CO)N(CC1CCCCC1)CCN2[C@H]3C[C@H](C4=CC(C(N)=O)=CC=C4)C[C@@H]2CC3.O=S(O)(O)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.