Fig. 1 · Structure
Documents & Downloads
AZ-GHS-22
GHS-R1a Inverse Agonist
AZ-GHS-22 is a potent inverse agonist targeting the growth hormone secretagogue receptor type 1a (GHS-R1a) with an IC50 of 0.77 nM. This compound exhibits significant inhibition of receptor activity, making it a valuable tool for research into metabolic regulation and appetite control. AZ-GHS-22 is particularly useful for studies focused on obesity and related disorders, enabling exploration of the physiological roles of GHS-R1a in non-central nervous system contexts.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inverse Agonist |
| CAS Number | 1143020-91-0 |
| Applications | GHS-R1a Inverse Agonist |
| Formula | C27H33ClN6O5S2 |
| Molecular Weight | 621.17 |
| SMILES | O=C(NC(NC1=NC2=CC=C(S(=O)(CCCN3CCN(C)CC3)=O)C=C2S1)=O)C4=CC(N5CCOCC5)=CC=C4Cl |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.