Fig. 1 · Structure
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BAY-252
BCAT1/2 Inhibitor
BAY-252 is a selective inhibitor of branched-chain amino acid transaminases 1 (BCAT1) and 2 (BCAT2), exhibiting IC50 values of 2 μM for both targets. This compound serves as a valuable chemical probe for investigating metabolic pathways involving branched-chain amino acids. BAY-252 is particularly relevant in cancer research, providing insights into tumor metabolism and potential therapeutic strategies.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 2639638-67-6 |
| Applications | BCAT1/2 Inhibitor |
| Formula | C22H14ClF3N2O3 |
| Molecular Weight | 446.81 |
| SMILES | CC(C=CC=C1)=C1OC2=C(Cl)C3=C(C=CC=C3)C(N4C(NC(C(F)(F)F)=CC4=O)=O)=C2 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.