BAY-8002

Catalog No.: A18611

MCT1 inhibitor

BAY-8002

BAY-8002 Chemical Structure

CAS NO. 724440-27-1

BAY-8002 is a potent, selective, orally active inhibitor of monocarboxylate transporter 1 (MCT1), with an IC50 of 85 nM in the MCT1-expressing DLD-1 cells, displays excellent selectivity against MCT4. Anti-tumor activity.

Availability: In stock

Package Price Qty
5 mg
$90.00
10 mg
$140.00
50 mg
$420.00
100 mg
$720.00
Custom Size Get quote

Free Overnight Delivery on orders over $500

Next day delivery by 10:00 a.m. Order now.

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

BAY-8002 is a potent, selective, orally active inhibitor of monocarboxylate transporter 1 (MCT1), with an IC50 of 85 nM in the MCT1-expressing DLD-1 cells, displays excellent selectivity against MCT4. Anti-tumor activity.
In vitro DMSO 73 mg/mL (175.54 mM)
Water Insoluble
Ethanol 25 mg/mL (60.12 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 24.05 mL 120.24 mL 240.47 mL
0.5 mM 4.81 mL 24.05 mL 48.09 mL
1 mM 2.4 mL 12.02 mL 24.05 mL
5 mM 0.48 mL 2.4 mL 4.81 mL

*The above data is based on the productmolecular weight 415.85. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A18611
Actions Inhibitor
CAS No. 724440-27-1
Formula C20H14ClNO5S
M. Wt 415.85
Solubility DMSO
Purity >98%
Synonyms BAY8002, BAY 8002
SMILES O=C(O)C1=CC=CC=C1NC(C2=CC(S(=O)(C3=CC=CC=C3)=O)=CC=C2Cl)=O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Product Tags

Product Tags

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy BAY-8002 | BAY-8002 Supplier | purchase | cost | manufacturer | order | distributor | buy 724440-27-1| 724440-27-1 Supplier | purchase 724440-27-1 | 724440-27-1 cost | 724440-27-1 manufacturer | order 724440-27-1 | 724440-27-1 distributor
Rewards