Fig. 1 · Structure
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BET-IN-6
PROTAC Ligand
BET-IN-6 is a high-affinity inhibitor targeting BRD2 and BRD4. As a key ligand for these bromodomain proteins, BET-IN-6 is utilized in the synthesis of the PROTAC BRD2/BRD4 degrader-1. Its application is significant in epigenetic research and protein degradation studies, making it a valuable tool for investigating cellular processes regulated by BRD2 and BRD4.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 2570470-39-0 |
| Applications | PROTAC Ligand |
| Formula | C22H20N2O6S |
| Molecular Weight | 440.47 |
| SMILES | O=C(O)CCC1=CC2=C(C=CC(N(C3=O)C)=C2C3=C1)NS(=O)(C4=CC=CC=C4OC)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.