BIM 21009

Catalog No.: A60761
LHRH/GnRH Receptor Antagonist
BIM 21009 is a potent LHRH/GnRH receptor antagonist, primarily targeting the gonadotropin-releasing hormone pathway. It demonstrates significant inhibitory effects on tumor growth, making it an essential tool for research in oncology and reproductive biology. BIM 21009 is valuable for studies focused on hormone-dependent cancers and the modulation of reproductive functions.
Grouped product items
Size Price Stock Qty
25mg
$1,275.00
In stock
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Bulk Discount
Free Delivery on orders over $500
Research use only. We do not sell to patients.

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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
DescriptionBIM 21009 is a potent LHRH/GnRH receptor antagonist, primarily targeting the gonadotropin-releasing hormone pathway. It demonstrates significant inhibitory effects on tumor growth, making it an essential tool for research in oncology and reproductive biology. BIM 21009 is valuable for studies focused on hormone-dependent cancers and the modulation of reproductive functions.
Product Information
Catalog NumA60761
FormulaC74H92ClN17O13
Molecular Weight1463.08
CAS Number106881-54-3
SequenceAc-{d-Nal}-{d-Cl-Phe}-{d-Phe}-Ser-Tyr-{d-Arg}-Phe-Arg-Pro-{d-Ala}-NH2
Sequence shorteningAc-{d-Nal}-{d-Cl-Phe}-{d-Phe}-SY-{d-Arg}-FRP-{d-Ala}-NH2
SMILESC([C@@H](NC([C@H](CC1=CC=CC=C1)NC([C@H](NC([C@H](CC2=CC=C(O)C=C2)NC([C@@H](NC([C@H](NC([C@@H](CC3=CC=C(Cl)C=C3)NC([C@@H](CC4=CC5=C(C=C4)C=CC=C5)NC(C)=O)=O)=O)CC6=CC=CC=C6)=O)CO)=O)=O)CCCNC(=N)N)=O)=O)CCCNC(=N)N)(=O)N7[C@H](C(N[C@@H](C(N)=O)C)=O)CCC7
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