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BJP-07-017-3

Pin1 Inhibitor

BJP-07-017-3 is a potent inhibitor of proline cis-trans isomerase (Pin1) with an IC50 of 9 nM. It covalently modifies the cysteine residue at position 113 of Pin1, causing significant conformational changes that impair its stability. This interaction leads to proteasome-mediated degradation of Pin1, making BJP-07-017-3 a valuable tool for investigating cellular processes regulated by Pin1. It is suitable for research applications focused on cancer and neurodegenerative diseases where Pin1 plays a critical role.

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Specifications

Manufacturer	Adooq Bioscience
Actions	Inhibitor
CAS Number	2468783-22-2
Applications	Pin1 Inhibitor
Formula	C₃₅H₄₅ClN₈O₆
Molecular Weight	709.23
SMILES	CN(C(CCl)=O)[C@H](C(N1CCCC[C@H]1C(N[C@H](C(N[C@@H](CCCNC(N)=O)C(N)=O)=O)CC2=CNC3=C2C=CC=C3)=O)=O)CC4=CC=CC=C4

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.