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BMS-863233, also known as XL-413, is an orally bioavailable cell division cycle 7 homolog (CDC7) kinase inhibitor with potential antineoplastic activity.
Targets
| Cdc7 | Pim1 | CK2 | ||
| 3.4 nM | 42 nM | 212 nM |
| In vitro | DMSO | 46 mg/mL heating (141.02 mM) | |
| Water | <1 mg/mL (<1 mM) | ||
| Ethanol | <1 mg/mL (<1 mM) | ||
|
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
|||
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 30.66 mL | 153.29 mL | 306.58 mL |
| 0.5 mM | 6.13 mL | 30.66 mL | 61.32 mL |
| 1 mM | 3.07 mL | 15.33 mL | 30.66 mL |
| 5 mM | 0.61 mL | 3.07 mL | 6.13 mL |
*The above data is based on the productmolecular weight 326.18. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Technical Details
| Catalog Num | A13677 |
|---|---|
| Actions | Inhibitor |
| M. Wt | 326.18 |
| Formula | C14H13Cl2N3O2 |
| Solubility | DMSO |
| Purity | >98% |
| Storage | at -20°C 3 years Powder |
| CAS No. | 1169562-71-3 |
| Synonyms | BMS-863233; BMS863233; BMS 863233; XL-413; XL413; XL 413 |
| SMILES | C1C[[email protected]](NC1)C2=NC(=O)C3=C(N2)C4=C(O3)C=CC(=C4)Cl.Cl |
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