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BRD4 ligand 15

BRD4 Ligand

BRD4 Ligand 15 is an alkyne-modified chalcone derivative that specifically targets the bromodomain-containing protein 4 (BRD4). This compound serves as a crucial building block for the synthesis of BRD4-targeting PROTACs, exemplified by TKP-5. Its application in research includes the study of BRD4-related pathways and the development of targeted protein degradation therapies.

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Specifications

Manufacturer	Adooq Bioscience
Actions	Ligand / Binder
CAS Number	3076613-24-3
Applications	BRD4 Ligand
Formula	C₂₅H₂₇NO₅
Molecular Weight	421.49
SMILES	O=C(C)NCCC1=C(C(/C=C/C2=CC=C(OCC#C)C=C2)=O)C=C(OCC)C(OC)=C1

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.