BRL-54443
Important Notice: For research use only. We do not sell to patients.
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Important Notice: For research use only. We do not sell to patients.
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Discription | BRL 54443 is a 5-HT1E and 5-HT1F receptor agonist with pKi of 8.7 and 9.25, respectively, with a weak binding affinity for 5-HT1A, 5-HT1B, 5-HT1D receptors. | ||
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Targets |
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Catalog Num | A15592 |
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Formula | C14H18N2O |
Molecular Weight | 230.31 |
CAS Number | 57477-39-1 |
SMILES | CN1CCC(CC1)C2=CNC3=C2C=C(C=C3)O |
Synonyms | BRL54443, BRL 54443 |
Storage | Store lyophilized at -20ºC, keep desiccated. |
In vitro (25°C) | DMSO | 40 mg/mL (173.68 mM) | |
Water | Insoluble | ||
Ethanol | 2 mg/mL (8.68 mM) | ||
In vivo | 30% propylene glycol, 5% Tween 80, 65% D5W | 28 mg/mL | |
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 43.42 mL | 217.1 mL | 434.2 mL |
0.5 mM | 8.68 mL | 43.42 mL | 86.84 mL |
1 mM | 4.34 mL | 21.71 mL | 43.42 mL |
5 mM | 0.87 mL | 4.34 mL | 8.68 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2