BRL-54443

Catalog No.: A15592
5-HT1E/5-HT1F receptor agonist
BRL 54443 is a 5-HT1E and 5-HT1F receptor agonist with pKi of 8.7 and 9.25, respectively, with a weak binding affinity for 5-HT1A, 5-HT1B, 5-HT1D receptors.
Grouped product items
Product Name Price Stock Qty
BRL-54443 10mg
$70.00
In stock
BRL-54443 25mg
$140.00
In stock
BRL-54443 100mg
$550.00
In stock
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Biological Activity
Discription BRL 54443 is a 5-HT1E and 5-HT1F receptor agonist with pKi of 8.7 and 9.25, respectively, with a weak binding affinity for 5-HT1A, 5-HT1B, 5-HT1D receptors.
Targets
Target Value
Product Information
Catalog Num A15592
Formula C14H18N2O
Molecular Weight 230.31
CAS Number 57477-39-1
SMILES CN1CCC(CC1)C2=CNC3=C2C=C(C=C3)O
Synonyms BRL54443, BRL 54443
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Solubility
In vitro (25°C) DMSO 40 mg/mL (173.68 mM)
Water Insoluble
Ethanol 2 mg/mL (8.68 mM)
In vivo 30% propylene glycol, 5% Tween 80, 65% D5W 28 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Preparing Stock Solutions
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 43.42 mL 217.1 mL 434.2 mL
0.5 mM 8.68 mL 43.42 mL 86.84 mL
1 mM 4.34 mL 21.71 mL 43.42 mL
5 mM 0.87 mL 4.34 mL 8.68 mL
Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

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