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Bromodomain IN-2

BD Inhibitor

Bromodomain IN-2 is a selective bromodomain (BD) inhibitor that targets key bromodomain-containing proteins involved in epigenetic regulation. It exhibits strong biological activity with KD values of 250 nM for BRD4(1), 420 nM for CBP, and 130 nM for BRPF1B, among others. Its antiproliferative properties make it a valuable tool in cancer research and the study of epigenetic modifications. Bromodomain IN-2 is suitable for applications exploring BD-dependent cellular processes and therapeutic interventions.

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Specifications

Manufacturer	Adooq Bioscience
Actions	Inhibitor
CAS Number	2445335-77-1
Applications	BD Inhibitor
Formula	C₁₆H₁₇ClN₂O
Molecular Weight	288.77
SMILES	O=C1C2=C(C)NC(C3=C(Cl)C=CC(N)=C3)=C2CCCC1

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.