Fig. 1 · Structure
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BU-E-75
H2 Receptor Agonist/α-adrenoceptor AntagonisT
BU-E-75 is a guanidine-based compound that acts as an H2 receptor agonist while also exhibiting antagonistic properties at postsynaptic α-adrenoceptors. This dual functionality allows BU-E-75 to induce relaxation in noradrenaline-precontracted vessels, making it a valuable tool for studying vascular responses and adrenergic signaling pathways. Its unique action profile is relevant for research in cardiovascular pharmacology and receptor biology.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Agonist |
| CAS Number | 114667-74-2 |
| Applications | H2 Receptor Agonist/α-adrenoceptor AntagonisT |
| Formula | C21H24F2N6 |
| Molecular Weight | 398.45 |
| SMILES | FC1=CC=C(C(CCNC(NCCCC2=CN=CN2)=N)C3=NC=CC=C3)C=C1F |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.