Fig. 1 · Structure
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CARM1-IN-3
CARM1 Inhibitor
CARM1-IN-3 is a selective inhibitor of the co-activator associated arginine methyltransferase 1 (CARM1), demonstrating an IC50 value of 0.07 µM for CARM1 and >25 µM for CARM3. This compound is valuable for studying the regulatory roles of CARM1 in gene expression and its impact on various biological processes. Research applications include investigating the function of arginine methylation in transcriptional regulation and exploring potential therapeutic targets in related diseases.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 912970-67-3 |
| Applications | CARM1 Inhibitor |
| Formula | C24H32N4O2 |
| Molecular Weight | 408.54 |
| SMILES | CNCCN1CCC(C2=CC3=C(N=C(C4=C(OC)C=CC=C4OC)N3)C(C)=C2)CC1 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.