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CaSR antagonist-1

CaSR Antagonist

CaSR antagonist-1 is a potent antagonist of the calcium-sensing receptor (CaSR) with an IC50 value of 50 nM. This compound is valuable for investigating disorders linked to abnormal bone and mineral homeostasis, including osteoporosis. Its ability to modulate CaSR activity makes it a useful tool in research exploring the pathways involved in calcium metabolism and skeletal health.

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Specifications

Manufacturer	Adooq Bioscience
Actions	Antagonist
CAS Number	1219811-83-2
Applications	CaSR Antagonist
Formula	C₂₉H₂₄FN₃O₂S
Molecular Weight	497.58
SMILES	O=C1C(C2=CC(C3=CC=CC=N3)=C(C)S2)=C(C)N=C(N1CCC4=CC=CC=C4)C5=C(O)C(F)=CC=C5

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.