Fig. 1 · Structure
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Cavα2δ-IN-1
Cavα2δ Inhibitor
Cavα2δ-IN-1 is a selective inhibitor of the Cavα2δ-1 voltage-gated calcium channel, exhibiting a Ki value of 6 nM, indicating strong affinity. This compound shows remarkable selectivity against Cavα2δ-2, with a Ki greater than 10,000 nM. Cavα2δ-IN-1 is utilized in research applications focused on neuropharmacology and pain management, providing insights into calcium signaling pathways and potential therapeutic interventions.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 2416957-09-8 |
| Applications | Cavα2δ Inhibitor |
| Formula | C18H27N5O |
| Molecular Weight | 329.44 |
| SMILES | O=C1C(C=NC=C2)=C2N=C([C@H](N3C[C@@H](C)NCC3)CCC)N1CC |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.