CB2R/5-HT1AR agonist 1 is a dual agonist targeting the CB2 receptor and the 5-HT1A receptor, displaying partial agonism at the former (EC50=479.6 nM) and full agonism at the latter (EC50=2.7 μM). This compound demonstrates significant anti-anxiety and anti-depressive effects, making it relevant for research in neurological and psychiatric applications. Additionally, it exhibits favorable pharmacokinetic properties, enhancing its potential as a therapeutic candidate.
CB2R/5-HT1AR agonist 1 is a dual agonist targeting the CB2 receptor and the 5-HT1A receptor, displaying partial agonism at the former (EC50=479.6 nM) and full agonism at the latter (EC50=2.7 μM). This compound demonstrates significant anti-anxiety and anti-depressive effects, making it relevant for research in neurological and psychiatric applications. Additionally, it exhibits favorable pharmacokinetic properties, enhancing its potential as a therapeutic candidate.
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