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CB2R/5-HT1AR agonist 1

CB2R/5-HT1AR Agonist

CB2R/5-HT1AR agonist 1 is a dual agonist targeting the CB2 receptor and the 5-HT1A receptor, displaying partial agonism at the former (EC50=479.6 nM) and full agonism at the latter (EC50=2.7 μM). This compound demonstrates significant anti-anxiety and anti-depressive effects, making it relevant for research in neurological and psychiatric applications. Additionally, it exhibits favorable pharmacokinetic properties, enhancing its potential as a therapeutic candidate.

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Specifications

Manufacturer	Adooq Bioscience
Actions	Agonist
CAS Number	2821085-76-9
Applications	CB2R/5-HT1AR Agonist
Formula	C₂₄H₃₃NO₃
Molecular Weight	383.52
SMILES	CCCCC1(C2=C(C(O)=C([C@H]3[C@@H](CCC(C)=C3)C(C)=C)C(O)=C2)C(N)=O)CC1

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.