Biological Activity
Centrinone (LCR-263) is a selective and reversible inhibitor of polo-like kinase 4 (PLK4) with a Ki of 0.16 nM.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 15.78 mL | 78.91 mL | 157.82 mL |
0.5 mM | 3.16 mL | 15.78 mL | 31.56 mL |
1 mM | 1.58 mL | 7.89 mL | 15.78 mL |
5 mM | 0.32 mL | 1.58 mL | 3.16 mL |
*The above data is based on the productmolecular weight 633.65. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Catalog Num | A20858 |
---|---|
Actions | Inhibitor |
CAS No. | 1798871-30-3 |
Formula | C26H25F2N7O6S2 |
M. Wt | 633.65 |
Purity | >98% |
Synonyms | LCR-263, LCR 263, LCR263 |
SMILES | FC(C([N+]([O-])=O)=CC=C1)=C1CS(C2=CC(F)=C(SC3=NC(NC4=NNC(C)=C4)=C(OC)C(N5CCOCC5)=N3)C=C2)(=O)=O |
Storage | Store lyophilized at -20ºC, keep desiccated. |
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