Centrinone

Catalog No.: A20858

PLK4 inhibitor

Centrinone

Centrinone Chemical Structure

CAS NO. 1798871-30-3

Centrinone (LCR-263) is a selective and reversible inhibitor of polo-like kinase 4 (PLK4) with a Ki of 0.16 nM.

Availability: In stock

Package Price Qty
5 mg
$130.00
10 mg
$223.00
50 mg
$662.00
100 mg
$1,325.00
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Biological Activity

Centrinone (LCR-263) is a selective and reversible inhibitor of polo-like kinase 4 (PLK4) with a Ki of 0.16 nM.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 15.78 mL 78.91 mL 157.82 mL
0.5 mM 3.16 mL 15.78 mL 31.56 mL
1 mM 1.58 mL 7.89 mL 15.78 mL
5 mM 0.32 mL 1.58 mL 3.16 mL

*The above data is based on the productmolecular weight 633.65. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A20858
Actions Inhibitor
CAS No. 1798871-30-3
Formula C26H25F2N7O6S2
M. Wt 633.65
Purity >98%
Synonyms LCR-263, LCR 263, LCR263
SMILES FC(C([N+]([O-])=O)=CC=C1)=C1CS(C2=CC(F)=C(SC3=NC(NC4=NNC(C)=C4)=C(OC)C(N5CCOCC5)=N3)C=C2)(=O)=O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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