Fig. 1 · Structure
Documents & Downloads
Cerlapirdine
5-HT6 Antagonist
Cerlapirdine is a selective and potent full antagonist of the 5-hydroxytryptamine 6 (5-HT6) receptor. This compound demonstrates significant biological activity in modulating neurotransmitter systems, making it a valuable reagent for studying neurodegenerative disorders, particularly Alzheimer's disease. Cerlapirdine's antagonistic properties facilitate research into cognitive functions and the underlying mechanisms associated with synaptic plasticity and memory.
In Stock
Free Aliquoting for Your Order
Tell us your preferred amount per vial. We’ll confirm the options.
Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 925448-93-7 |
| Applications | 5-HT6 Antagonist |
| Formula | C22H23N3O3S |
| Molecular Weight | 409.50 |
| Synonyms | SAM-531; PF-05212365 |
| SMILES | O=S(C1=NNC2=C1C=C(OCCCN(C)C)C=C2)(C3=C4C=CC=CC4=CC=C3)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.