Fig. 1 · Structure
Documents & Downloads
CGP 20712 A
β1-Adrenoceptor Antagonist
CGP 20712 A is a highly selective β1-adrenoceptor antagonist, demonstrating an IC50 of 0.7 nM and approximately 10,000-fold selectivity over β2-adrenoceptors. This compound is primarily utilized in research applications investigating cardiovascular physiology and pharmacology. Its potent inhibition of β1-adrenoceptor activity makes it a valuable tool for studying the role of β1-adrenergic signaling in various biological processes.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 105737-62-0 |
| Applications | β1-Adrenoceptor Antagonist |
| Formula | C24H29F3N4O8S |
| Molecular Weight | 590.57 |
| Synonyms | CGP 20712 mesylate |
| SMILES | O=C(N)C1=CC(OCCNCC(O)COC2=CC=C(C3=NC(C(F)(F)F)=CN3C)C=C2)=CC=C1O.CS(=O)(O)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.