Fig. 1 · Structure
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CGP 20712
β1-Adrenoceptor Antagonist
CGP 20712 is a selective β1-adrenoceptor antagonist with a Ki value of 0.3 nmol/L. Its primary mechanism of action involves competitively binding to β1-receptors, effectively inhibiting the positive chronotropic effects induced by adrenaline and noradrenaline. CGP 20712 is utilized in research to study cardiovascular function and the role of β1-adrenoceptors in various physiological and pathological conditions.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 137888-49-4 |
| Applications | β1-Adrenoceptor Antagonist |
| Formula | C23H25F3N4O5 |
| Molecular Weight | 494.46 |
| SMILES | O=C(N)C1=CC(OCCNCC(O)COC2=CC=C(C3=NC(C(F)(F)F)=CN3C)C=C2)=CC=C1O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.