CHS-828 (GMX1778)

Catalog No.: A12515

NAMPT inhibitor

CHS-828 (GMX1778) Chemical Structure

CAS NO. 200484-11-3

CHS-828 is a potent inhibitor of NAD+ biosynthesis enzyme NAMPT with IC50 <25 nM.

Availability: In stock

Package Price Qty
5 mg
$50.00
10 mg
$70.00
25 mg
$150.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

CHS-828 is a potent inhibitor of NAD+ biosynthesis enzyme NAMPT with IC50 <25 nM.
Targets
NAMPT NAMPT
25 nM120 nM(Kd)
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 26.89 mL 134.46 mL 268.92 mL
0.5 mM 5.38 mL 26.89 mL 53.78 mL
1 mM 2.69 mL 13.45 mL 26.89 mL
5 mM 0.54 mL 2.69 mL 5.38 mL

*The above data is based on the productmolecular weight 371.86. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A12515
Actions Inhibitor
M. Wt 371.86
Formula C19H22ClN5O
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 200484-11-3
Synonyms GMX1778, GMX-1778, GMX 1778, CHS828, CHS 828
SMILES ClC1=CC=C(OCCCCCC/N=C(\N=C2C=CNC=C/2)NC#N)C=C1

Product Tags

Product Tags

Other people marked this product with these tags:

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy CHS-828 (GMX1778) | CHS-828 (GMX1778) Supplier | purchase CHS-828 (GMX1778) | CHS-828 (GMX1778) cost | CHS-828 (GMX1778) manufacturer | order CHS-828 (GMX1778) | CHS-828 (GMX1778) distributor | buy 200484-11-3| 200484-11-3 Supplier | purchase 200484-11-3 | 200484-11-3 cost | 200484-11-3 manufacturer | order 200484-11-3 | 200484-11-3 distributor
Rewards