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$0.00 Biological Activity
Cilengitide is a cyclic Arg-Gly-Asp peptide with potential antineoplastic activity. Cilengitide binds to and inhibits the activities of the alpha(v)beta(3) and alpha(v)beta(5) integrins, thereby inhibiting endothelial cell-cell interactions, endothelial cell-matrix interactions, and angiogenesis.
Targets
| αvβ3 receptor (Cell-free assay) | αvβ5 receptor (Cell-free assay) | |||
| 4.1 nM | 79 nM |
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 14.23 mL | 71.15 mL | 142.31 mL |
| 0.5 mM | 2.85 mL | 14.23 mL | 28.46 mL |
| 1 mM | 1.42 mL | 7.12 mL | 14.23 mL |
| 5 mM | 0.28 mL | 1.42 mL | 2.85 mL |
*The above data is based on the productmolecular weight 702.7. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A12371 |
|---|---|
| Actions | Inhibitor |
| M. Wt | 702.7 |
| Formula | C29H41N8O9F3 |
| Solubility | DMSO |
| Purity | >98% |
| Storage | at -20°C 3 years Powder |
| CAS No. | 199807-35-7 |
| Synonyms | EMD 12197,EMD-85189,EMD-121974,NSC-707544,D03497 |
| SMILES | CC(C)[[email protected]]1C(=O)N[[email protected]](C(=O)NCC(=O)N[[email protected]](C(=O)N[[email protected]@H](C(=O)N1C)Cc2ccccc2)CC(=O)O)CCCNC(=N)N.C(=O)(C(F)(F)F)O |
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