Fig. 1 · Structure
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CINPA1
CAR Inhibitor
CINPA1 is a potent and selective inhibitor of the constitutive androstane receptor (CAR), specifically inhibiting its activity without activating the pregnane X receptor (PXR). With an IC50 of approximately 70 nM, CINPA1 effectively reduces CAR-mediated transcriptional activity. This compound serves as a valuable tool for investigating the physiological and pathological roles of CAR in various biological processes.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 102636-74-8 |
| Applications | CAR Inhibitor |
| Formula | C23H29N3O3 |
| Molecular Weight | 395.49 |
| SMILES | CCN(CC)CC(N1C2=CC(NC(OCC)=O)=CC=C2CCC3=C1C=CC=C3)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.