Fig. 1 · Structure
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Cipralisant (enantiomer)
H3 Receptor Antagonist
Cipralisant (enantiomer) is a potent and selective antagonist of the histamine H3 receptor, demonstrating a high affinity binding with a rat Ki value of 0.47 nM. This compound serves as a valuable tool in the study of H3 receptor-mediated pathways, offering insights into neurological functions and disorders. Additionally, Cipralisant (enantiomer) features an alkyne functional group, enabling its use in click chemistry applications, particularly in copper-catalyzed azide-alkyne cycloaddition (CuAAc) reactions for bioconjugation purposes.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 223420-11-9 |
| Applications | H3 Receptor Antagonist |
| Formula | C14H20N2 |
| Molecular Weight | 216.32 |
| Synonyms | GT-2331 (enantiomer) |
| SMILES | CC(C)(C)CCC#C[C@@H]1[C@@H](C2=CN=CN2)C1 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.