Cisapride

Catalog No.: A21340

hERG potassium channel inhibitor

Cisapride

Cisapride Chemical Structure

CAS NO. 81098-60-4

Cisapride(R 51619) is a nonselective 5-HT4 receptor agonist, it is also a potent hERG potassium channel inhibitor.

Availability: In stock

Package Price Qty
10 mg
$65.00
25 mg
$130.00
50 mg
$223.00
100 mg
$382.00
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Biological Activity

Cisapride(R 51619) is a nonselective 5-HT4 receptor agonist, it is also a potent hERG potassium channel inhibitor.
In vitro DMSO 83 mg/mL (178.13 mM)
Water Insoluble
Ethanol Insoluble
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 21.46 mL 107.31 mL 214.62 mL
0.5 mM 4.29 mL 21.46 mL 42.92 mL
1 mM 2.15 mL 10.73 mL 21.46 mL
5 mM 0.43 mL 2.15 mL 4.29 mL

*The above data is based on the productmolecular weight 465.95. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21340
Actions Inhibitor
CAS No. 81098-60-4
Formula C23H29ClFN3O4
M. Wt 465.95
Purity >98%
Synonyms R 51619
SMILES ClC1=C(N)C=C(OC)C(C(N[[email protected]]2[[email protected]@H](OC)CN(CCCOC3=CC=C(F)C=C3)CC2)=O)=C1.[relative stereochemistry]
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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