Fig. 1 · Structure
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Conivaptan hydrochloride
Vasopressin Receptor Antagonist
Conivaptan hydrochloride is a selective non-peptide antagonist of the vasopressin receptors, specifically targeting the V1A and V2 subtypes. With Ki values of 0.48 nM and 3.04 nM for the rat liver V1A receptor and rat kidney V2 receptor, respectively, it effectively inhibits vasopressin-mediated responses. This compound is primarily applied in research related to fluid balance disorders and the investigation of vasopressin receptor signaling pathways.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 168626-94-6 |
| Applications | Vasopressin Receptor Antagonist |
| Formula | C32H27ClN4O2 |
| Molecular Weight | 535.04 |
| Synonyms | YM 087 |
| SMILES | O=C(C1=CC=CC=C1C2=CC=CC=C2)NC3=CC=C(C(N4CCC(N=C(C)N5)=C5C6=CC=CC=C64)=O)C=C3.Cl |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.