CP-601927 is a selective partial agonist of the α4β2 nicotinic acetylcholine receptor (nAChR), exhibiting a Ki value of 1.2 nM and an EC50 of 2.6 μM. This compound demonstrates effective brain penetration and possesses antidepressant-like properties, making it a valuable tool in neurological research. Its modulation of nAChR activity is relevant for studies exploring neuropsychiatric disorders and the underlying mechanisms of depression.
CP-601927 is a selective partial agonist of the α4β2 nicotinic acetylcholine receptor (nAChR), exhibiting a Ki value of 1.2 nM and an EC50 of 2.6 μM. This compound demonstrates effective brain penetration and possesses antidepressant-like properties, making it a valuable tool in neurological research. Its modulation of nAChR activity is relevant for studies exploring neuropsychiatric disorders and the underlying mechanisms of depression.
This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:
