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$0.00 Biological Activity
CPI-360 is a selective EZH2 inhibitor with IC50 values of 0.5 and 2.5 nM for wild-type EZH2 and Y641N mutant EZH2, respectively.
Targets
| EZH2 | ||||
| 0.25 nM |
| In vitro (25°C) | DMSO | Warmed: 18 mg/mL (41.14 mM) | |
| Water | Insoluble | ||
| Ethanol | Warmed: 16 mg/mL (36.57 mM) | ||
| In vivo | 10% DMSO+60% PEG 400+ddH2O | 19 mg/mL | |
|
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
|||
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 22.86 mL | 114.28 mL | 228.56 mL |
| 0.5 mM | 4.57 mL | 22.86 mL | 45.71 mL |
| 1 mM | 2.29 mL | 11.43 mL | 22.86 mL |
| 5 mM | 0.46 mL | 2.29 mL | 4.57 mL |
*The above data is based on the productmolecular weight 437.53. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A15908 |
|---|---|
| Actions | Inhibitor |
| CAS No. | 1802175-06-9 |
| Formula | C25H31N3O4 |
| M. Wt | 437.53 |
| Solubility | DMSO |
| Purity | >98% |
| Synonyms | CPI360, CPI 360 |
| SMILES | CC(N1)=CC(OC)=C(CNC(C2=C(C)N([[email protected]](C)C3CCOCC3)C4=C2C=CC=C4)=O)C1=O |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
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