CPI-360

Catalog No.: A15908

EZH1 inhibitor

CPI-360 Chemical Structure

CAS NO. 1802175-06-9

CPI-360 is a potent, selective,and SAM-competitive EZH1 inhibitor with IC50 of 102.3 nM, >100-fold selectivity over other methyltransferases.

Availability: In stock

Package Price Qty
5 mg
$140.00
10 mg
$195.00
25 mg
$420.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

CPI-360 is a potent, selective,and SAM-competitive EZH1 inhibitor with IC50 of 102.3 nM, >100-fold selectivity over other methyltransferases.
Targets
EZH1
102.3 nM
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 22.86 mL 114.28 mL 228.56 mL
0.5 mM 4.57 mL 22.86 mL 45.71 mL
1 mM 2.29 mL 11.43 mL 22.86 mL
5 mM 0.46 mL 2.29 mL 4.57 mL

*The above data is based on the productmolecular weight 437.53. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15908
Actions Inhibitor
M. Wt 437.53
Formula C25H31N3O4
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1802175-06-9
Synonyms CPI360, CPI 360
SMILES CC(N1)=CC(OC)=C(CNC(C2=C(C)N([[email protected]](C)C3CCOCC3)C4=C2C=CC=C4)=O)C1=O

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