Fig. 1 · Structure
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CPSA
AKR1C1 Inhibitor
CPSA is a potent and competitive inhibitor of 20α-hydroxysteroid dehydrogenase (AKR1C1), with a Ki value of 0.86 nM. This compound demonstrates significant biological activity, making it a valuable tool for investigating therapeutic avenues in lung and endometrial cancers, as well as conditions related to premature birth and neuronal disorders. CPSA's selective inhibition of AKR1C1 positions it as an important reagent for studying the biochemical pathways involved in these diseases.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 1038713-54-0 |
| Applications | AKR1C1 Inhibitor |
| Formula | C13H9ClO3 |
| Molecular Weight | 248.66 |
| SMILES | O=C(C1=CC(C2=CC=CC=C2)=CC(Cl)=C1O)O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.