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CX3CR1-IN-2

CX3CR1 Inhibitor

CX3CR1-IN-2 is a selective inhibitor of CX3CR1, demonstrating an IC50 of 0.04 μM. This compound effectively disrupts the binding of CX3CR1 to its ligand, fractalkine (CX3CL1). CX3CR1-IN-2 is valuable for studying cardiovascular diseases, including heart failure and cardiomyopathy, providing insights into the underlying mechanisms and potential therapeutic targets in these conditions.

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Specifications

Manufacturer	Adooq Bioscience
Actions	Inhibitor
CAS Number	3105688-14-7
Applications	CX3CR1 Inhibitor
Formula	C₁₉H₂₄F₃N₅O₄S₂
Molecular Weight	507.55
SMILES	FC(F)(F)C(C=CC=C1)=C1C(CSC2=NC(NS(C)(=O)=O)=NC(N[C@@H](CO)CC(C)C)=N2)=O

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.