Fig. 1 · Structure
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cyclo(RLsKDK)
ADAM8 Inhibitor
Cyclo(RLsKDK) is a potent inhibitor of the metalloproteinase ADAM8, exhibiting an IC50 value of 182 nM. This compound demonstrates significant anti-inflammatory properties and may serve as a valuable tool in the study of inflammatory diseases and cancer progression. Its selective inhibition of ADAM8 positions cyclo(RLsKDK) as a promising candidate for further research in therapeutic applications targeting these pathways.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 1975145-82-4 |
| Applications | ADAM8 Inhibitor |
| Formula | C31H57N11O9 |
| Molecular Weight | 727.85 |
| Synonyms | BK-1361 |
| SMILES | C(CCNC(=N)N)[C@@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](CO)NC(=O)[C@H](CC(C)C)NC1=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.