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D4R antagonist-1

D4R Antagonist

D4R antagonist-1 is a selective antagonist of the dopamine D4 receptor (D4R) with an IC50 of 6.87 µM. This compound exhibits significant potential for use in research related to neurological disorders, including Parkinson's disease. Its ability to modulate D4R activity makes it a valuable tool for investigating the role of dopamine signaling in various physiological and pathological processes.

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Specifications

Manufacturer	Adooq Bioscience
Actions	Antagonist
CAS Number	2846077-19-6
Applications	D4R Antagonist
Formula	C₂₁H₂₅F₂NO₂
Molecular Weight	361.43
SMILES	COC1=CC=C(C=C1F)CN2CCC[C@@H](C2)OCC3=CC(C)=C(C=C3)F

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.