Dersimelagon phosphate is a selective melanocortin 1 receptor (MC1R) agonist, exhibiting EC50 values of 8.16, 3.91, 1.14, and 0.251 nM for human, cynomolgus monkey, mouse, and rat MC1R, respectively. This compound demonstrates significant affinity for both hMC1R and hMC4R, with Ki values of 2.26 and 32.9 nM, respectively. Dersimelagon phosphate is utilized in research investigating skin pigmentation mechanisms and related biological processes.
Dersimelagon phosphate is a selective melanocortin 1 receptor (MC1R) agonist, exhibiting EC50 values of 8.16, 3.91, 1.14, and 0.251 nM for human, cynomolgus monkey, mouse, and rat MC1R, respectively. This compound demonstrates significant affinity for both hMC1R and hMC4R, with Ki values of 2.26 and 32.9 nM, respectively. Dersimelagon phosphate is utilized in research investigating skin pigmentation mechanisms and related biological processes.
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