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Biological Activity
Desmethyl-VS-5584 is a demethyl analogue of VS-5584, which is a novel and highly selective PI3K/mTOR kinase inhibitor for the treatment of cancer.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 29.38 mL | 146.89 mL | 293.78 mL |
| 0.5 mM | 5.88 mL | 29.38 mL | 58.76 mL |
| 1 mM | 2.94 mL | 14.69 mL | 29.38 mL |
| 5 mM | 0.59 mL | 2.94 mL | 5.88 mL |
*The above data is based on the productmolecular weight 340.391. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A10900 |
|---|---|
| Actions | Inhibitor |
| CAS No. | 1246535-95-4 |
| Formula | C16H20N8O |
| M. Wt | 340.391 |
| Purity | >98% |
| Synonyms | Desmethyl-VS-5584, Desmethyl-VS5584 |
| SMILES | NC1=NC=C(C2=C3N=CN(C(C)C)C3=NC(N4CCOCC4)=N2)C=N1 |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
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