Fig. 1 · Structure
Documents & Downloads
DG051 free acid
LTA4H Inhibitor
DG051 free acid is a potent inhibitor of leukotriene A4 hydrolase (LTA4H), exhibiting a Kd value of 26 nM. Its high water solubility (exceeding 30 mg/mL) and oral bioavailability (greater than 80% across multiple species) make it a valuable tool in biochemical studies. DG051 free acid is particularly applicable in research investigating myocardial infarction and stroke, providing insights into the modulation of inflammatory pathways associated with these conditions.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 929916-05-2 |
| Applications | LTA4H Inhibitor |
| Formula | C21H24ClNO4 |
| Molecular Weight | 389.87 |
| SMILES | ClC(C=C1)=CC=C1OC(C=C2)=CC=C2OC[C@H]3N(CCC3)CCCC(O)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.