Fig. 1 · Structure
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DGAT-1 inhibitor 3
DGAT-1 Inhibitor
DGAT-1 Inhibitor 3 is a selective inhibitor of diacylglycerol O-acyltransferase 1 (DGAT-1), exhibiting a potent inhibitory effect with an IC50 value of 0.038 µM. This compound is relevant for studies investigating lipid metabolism and has significant potential in obesity and diabetes research. Its activity can facilitate the understanding of DGAT-1's role in metabolic disorders and aid in the development of therapeutic strategies for associated diseases.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 1231243-91-6 |
| Applications | DGAT-1 Inhibitor |
| Formula | C21H20F3N3O3 |
| Molecular Weight | 419.40 |
| SMILES | O=C(C1=C(C(F)(F)F)OC(C2=CC=CC=C2)=N1)NC3=CC=C(N(CCOC)C)C=C3 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.