Fig. 1 · Structure
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DRAK1/2-IN-1
DRAK1/2 Inhibitor
DRAK1/2-IN-1 is a potent dual inhibitor of DRAK1 and DRAK2, exhibiting Kd values of 1 μM and 6 μM, respectively. This compound selectively targets DRAK family kinases, playing a crucial role in cell survival and apoptosis regulation. Its application extends to research on cancer biology, neurodegenerative diseases, and other conditions associated with dysregulated kinase activity.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 1629227-34-4 |
| Applications | DRAK1/2 Inhibitor |
| Formula | C22H24N2O3S |
| Molecular Weight | 396.50 |
| SMILES | O=C(C1CCCCC1)NC2=CSC3=NC=C(C4=CC(OC)=C(OC)C=C4)C=C32 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.