Fig. 1 · Structure
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(E/Z)-Endoxifen
Cytochrome P450 Inhibitor
Endoxifen is an active metabolite of tamoxifen that primarily targets and modulates the estrogen receptor, exhibiting higher binding affinity and specificity. In addition, it functions as a cytochrome P450 inhibitor, effectively inhibiting aromatase activity. Due to its unique profile, Endoxifen is valuable for research applications in breast cancer biology and therapeutic development.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 110025-28-0 |
| Applications | Cytochrome P450 Inhibitor |
| Formula | C25H27NO2 |
| Molecular Weight | 373.49 |
| SMILES | CC/C(C1=CC=CC=C1)=C(C2=CC=C(O)C=C2)/C3=CC=C(OCCNC)C=C3 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.