Fig. 1 · Structure
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E7016
PARP Inhibitor
E7016 is a potent orally bioavailable inhibitor of PARP (Poly(ADP-ribose) polymerase). By inhibiting DNA repair mechanisms, E7016 enhances the radiosensitivity of tumor cells both in vitro and in vivo, making it a promising candidate for cancer therapeutics. This compound is useful in research applications focused on cancer treatment strategies involving DNA damage response and repair pathways.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 902128-92-1 |
| Applications | PARP Inhibitor |
| Formula | C20H19N3O3 |
| Molecular Weight | 349.38 |
| Synonyms | GPI 21016 |
| SMILES | O=C1NN=C2C3=C1C=CC=C3OC4=CC=C(CN5CCC(O)CC5)C=C42 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.