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EA-B2L

GSTP Degrader

EA-B2L is a potent glutathione S-transferase P (GSTP) degrader, exhibiting a DC50 value of 48 μM. This compound is a Boc2Lys-linked Ethacrynic acid derivative, making it a valuable tool for studying GSTP-related pathways. Its ability to selectively degrade GSTP contributes to advancements in cancer research, allowing for the exploration of therapeutic strategies targeting GSTP expression and function.

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Specifications

Manufacturer	Adooq Bioscience
Actions	Degrader
CAS Number	1354444-72-6
Applications	GSTP Degrader
Formula	C₃₅H₅₄Cl₂N₄O₈
Molecular Weight	729.73
SMILES	CCC(C(C1=C(C(Cl)=C(C=C1)OCC(NCCCCCCNC([C@H](CCCCNC(OC(C)(C)C)=O)NC(OC(C)(C)C)=O)=O)=O)Cl)=O)=C

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.