Fig. 1 · Structure
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Elarofiban
Fibrinogen Receptor Antagonist
Elarofiban is a nonpeptide, orally active antagonist of the fibrinogen receptor αIIbβ3 (GPIIb/IIIa), exhibiting an IC50 of 0.15 nM. This compound disrupts platelet aggregation, making it a valuable tool for investigating platelet-mediated thrombotic disorders. Elarofiban's mechanism of action supports research into cardiovascular diseases and the development of antithrombotic therapies.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 198958-88-2 |
| Applications | Fibrinogen Receptor Antagonist |
| Formula | C22H32N4O4 |
| Molecular Weight | 416.51 |
| Synonyms | RWJ-53308 |
| SMILES | O=C(N[C@H](C1=CN=CC=C1)CC(O)=O)[C@H]2CN(CCC2)C(CCC3CCNCC3)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.