Eletriptan-d5 is a deuterium-labeled analog of Eletriptan, a highly selective and orally active agonist for the serotonin 5-HT1B and 5-HT1D receptors, exhibiting pKi values of 8.0 and 8.9, respectively. This compound demonstrates inhibitory effects on neurogenic inflammation markers in preclinical models, particularly in rats. Eletriptan-d5 is valuable for research applications focused on migraine pathophysiology and the pharmacological profiling of serotonin receptor interactions.
Eletriptan-d5 is a deuterium-labeled analog of Eletriptan, a highly selective and orally active agonist for the serotonin 5-HT1B and 5-HT1D receptors, exhibiting pKi values of 8.0 and 8.9, respectively. This compound demonstrates inhibitory effects on neurogenic inflammation markers in preclinical models, particularly in rats. Eletriptan-d5 is valuable for research applications focused on migraine pathophysiology and the pharmacological profiling of serotonin receptor interactions.
This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:
