Fig. 1 · Structure
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Enerisant
H3 Receptor Antagonist
Enerisant is a highly selective and competitive antagonist/inverse agonist of the histamine H3 receptor, exhibiting IC50 values of 2.89 nM for human receptors and 14.5 nM for rat receptors. Its oral bioavailability makes it a valuable tool for research focused on neurological disorders and cognitive enhancement. Enerisant is useful in studies investigating the role of histamine H3 receptors in neurotransmission, and it may facilitate the development of novel therapeutic strategies for related conditions.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 1152747-82-4 |
| Applications | H3 Receptor Antagonist |
| Formula | C22H30N4O3 |
| Molecular Weight | 398.50 |
| Synonyms | TS-091 |
| SMILES | O=C(C1=CN(C2=CC=C(OCCCN3[C@H](C)CCC3)C=C2)N=C1)N4CCOCC4 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.