Fig. 1 · Structure
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Enpp-1-IN-13
ENPP Inhibitor
Enpp-1-IN-13 is a selective inhibitor of ectonucleotide pyrophosphatase/phosphodiesterase (ENPP), demonstrating IC50 values of 1.29 μM against ENPP1 and 20.2 μM against ENPP3. This compound exhibits significant anticancer activity, making it a valuable tool for research on cancer biology and therapeutic development. Its inhibition of ENPP enzymes may provide insights into metabolic regulation and potential treatment pathways for various cancers.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 2417022-19-4 |
| Applications | ENPP Inhibitor |
| Formula | C28H22ClN5OS |
| Molecular Weight | 512.03 |
| SMILES | S=C(NC1=CC=CC=C1)NC2=CC=CC(N3N=C(C4=CC=C(OC)C(Cl)=C4)C(C5=CC=NC=C5)=C3)=C2 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.