Fig. 1 · Structure
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Enpp-1-IN-2
ENPP1 Inhibitor
Enpp-1-IN-2 is a potent inhibitor of ectonucleotide pyrophosphatase/phosphodiesterase 1 (ENPP1), exhibiting IC50 values of 0.26 μM, 0.48 μM, and 2.0 μM determined through TG-mAMP, pNP-TMP, and ATP assays, respectively. This compound provides a valuable tool for studying ENPP1 activity and its associated biological pathways. Its application in research may contribute to a better understanding of various physiological processes and disease mechanisms related to purinergic signaling and ecto-nucleotide metabolism.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 2378640-92-5 |
| Applications | ENPP1 Inhibitor |
| Formula | C15H18N6 |
| Molecular Weight | 282.34 |
| SMILES | CC1=NC2=NC=NN2C(N(C)C)=C1CC3=CC=CC(N)=C3 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.