Fig. 1 · Structure
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Enpp-1-IN-21
ENPP1 Inhibitor
Enpp-1-IN-21 is a potent inhibitor of ecto-nucleotide pyrophosphatase/phosphodiesterase 1 (ENPP1), demonstrating an IC50 of 0.45 μM against ENPP1 and 0.19 μM against ENPP3. This compound is valuable for studying the enzymatic regulation of nucleotide metabolism and is particularly relevant in research focused on cancer cell signaling and metabolic disorders. Its specificity towards ENPP1 positions it as a key tool for elucidating the physiological roles of this enzyme in various biological systems.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 2803505-78-2 |
| Applications | ENPP1 Inhibitor |
| Formula | C21H16F3NO5S |
| Molecular Weight | 451.42 |
| SMILES | O=C(C1=CC=C(C)C=C1)NC2=CC=C(C=C2)OS(=O)(C3=CC=C(C=C3)OC(F)(F)F)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.