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Ep300/CREBBP-IN-4

Ep300/CREBBP Inhibitor

Ep300/CREBBP-IN-4 is a potent inhibitor of Ep300 and CREBBP, with IC50 values of 0.024 μM and 0.064 μM, respectively. This compound is valuable for investigating the role of these acetyltransferases in cancer biology and related therapeutic avenues. Its ability to selectively inhibit Ep300 and CREBBP makes it a useful tool for cancer research applications.

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Specifications

Manufacturer	Adooq Bioscience
Actions	Inhibitor
CAS Number	2259641-42-2
Applications	Ep300/CREBBP Inhibitor
Formula	C₂₃H₂₂F₃N₅O₃
Molecular Weight	473.45
SMILES	O=C(N1[C@H](C[C@H](C1)F)C(NC2=CC=C(NN=C3)C3=N2)=O)C4(C5=CC=C(C=C5)OC)CC(F)(C4)F

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.